Raw Harshen HCL Mawasa (1431697-94-7)
Raw Lorcaserin HCL foda (1431697-94-7) Bayani
Product Name | Raw Lorcaserin Hydrochloride foda |
Chemical Name | raw Lorcaserin HCL powder,Lorcaserin |
Brand Name | BELVIQ |
Drug Class | 5-HT2C mai karɓar mai karɓa |
CAS Number | 1431697-94-7 |
InChIKey | ITIHHRMYZPNGRC-QRPNPIFTSA-N |
Kwayoyin halitta FƘararraki | C11H15Cl2N |
Kwayoyin halitta Wtakwas | 232.15 |
Monoisotopic Mass | 231.058154899 |
Gyarawa Point | Babu bayanai akwai |
Freezing Point | Babu bayanai akwai |
Half Half-Life | Rabin rabi na lorcaserin ne kamar 11 hours.Lorcaserin foda an kawar da farko a cikin fitsari (92%) da kuma a cikin feces (2.2%) |
Launi | White foda |
solubility | Rashin ruwa na ruwa: 0.0709 mg / ml |
Storage Taikin zafi | -20 ° C. |
Aaikace-aikace | Serotonin 2C (HT2C) receptor agonist for nauyi asara.Decreases food consumption and promotes satiety centrally |
Raw Lorcaserin Hcl foda (1431697-94-7) Bayani
Raw Lorcaserin hydrochloride powder is a hydrochloride obtained by reaction of lorcaserin powder with one equivalent of hydrochloric acid. Used as an anti-obesity drug. Lorcaserin hydrochloride is a 5HT2c receptor agonist indicated for use in adults with a BMI ≥30, or those with a BMI ≥27 and at least one weight-related condition like hypertension, type 2 diabetes or dyslipidemia.Lorcaserin Hydrochloride powder works by suppressing appetite and induces a feeling of satiety, and is thought to avoid the precipitation of cardiac valvular disease associated with activation of 5-HT2B receptors, the area of the brain known to play a major role in regulating hunger and food intake. By activating these receptors, Lorcaserin hydrochloride powder may decrease food consumption by decreasing appetite and making a person feel full even after eating less food than usual. was approved today by the FDA in a landmark decision after 2 years of scrutiny.
Ana ba da alamar samfurori mai gina jiki a cikin jiki mai saukin rage yawan karancin jiki (BMI na 30 kg / m2 ko mafi girma) kuma babba babba (BMI na 27 kg / m2 ko mafi girma) tare da akalla nau'in sharaɗɗa masu dangantaka da nauyi.
An yi amfani da man fetur na lantarki na Lorcaserin tare da abinci da motsa jiki don bi da kiba. Ana amfani da shi a wasu lokuta da kiba wanda zai iya dangantaka da ciwon sukari, high cholesterol, ko cutar hawan jini.
Lorcaserin hydrochloride ba za ta bi da wani yanayin lafiya ba (kamar cututtukan zuciya, ciwon sukari, hawan jini). Ci gaba da shan wasu magunguna da likitanku ya tsara don biyan waɗannan yanayi.
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Kodayake ba'a san ainihin ainihin aikin ba, an yi imanin ya ƙunshi zaɓin zaɓi na masu karɓa na 5-HT2C a cikin ƙananan neorexigenic pro-opiomelanocortin ne a cikin tsakiya na hypothalamus. Wannan yana haifar da rage yawan abincin abinci da rashin jin daɗi ta hanyar inganta sakin hormone na alpha-melanocortin, wanda ke aiki akan masu karɓa na melanocortin-4.
Lorcaserin hydrochloride foda yana aiki ta hanyar sarrafa abinci - musamman ta hanyar kunna masu karɓar kwakwalwa don serotonin, wani ɗan kwayar cutar da ke haifar da jin daɗi da gamsuwa. Samun abinci yana sarrafawa ne ta hanyar cibiyar satiety, wanda ke cikin kwayar iska ta hypothalamus da cibiyar yunwa da ke cikin hypothalamus na gefe. Ayyuka iri-iri daga manyan cibiyoyi da hanyoyin hanji suna haɗuwa a tsakiya, inda nau'ikan nau'ikan jijiyoyi biyu masu sarrafa abincin suke. Da fari dai, ƙungiyar mai cin abinci mai haɓaka abinci mai haɓaka furotin da ke da alaƙa da agouti da neuropeptide Y; kuma na biyu, ƙungiyar hana cin abinci da ke ƙunshe da hodar iblis da amphetamine da aka tsara kwafi (CART) da ƙwayoyin cuta na pro-opiomelanocortin (POMC). POMC ya ƙunshi masu karɓar 5-HT 2C, wanda lokacin da aka kunna su yana fitar da hawan mai kara alpha-melanocyte (alfa-MSH). Paraaƙarin tsakiya yana ƙunshe da masu karɓar melanocyte 4 (MC4R) wanda ke hana ci abinci a cikin allurai na kwayoyi lorcaserin hydrochloride foda yana aiki azaman mai zaɓin 5-HT 2C agonist akan ƙwayoyin POMC, wanda hakan yana haifar da sakin alfa MSH. Arin alfa MSH yana aiki akan MC4R a cikin tsakiya mai mahimmanci a cikin hypothalamus, wanda ke haifar da rage yawan ci. A cikin magungunan asibiti, lorcaserin hydrochlorider yana aiki akan 5-HT 2B da masu karɓa na 5-HT 2A.
amfanin na ƙwayar Lorcaserin Hcl (1431697-94-7)
- Lorcaserin HCL powder is a selective 5-HT2C receptor agonist that is thought to decrease food intake through the central POMC system. Lorcaserin HCL amfanin foda:
- Ana amfani da furotin na Cizon Lakaci tare da abinci da motsa jiki don bi da kiba.
- Ana yin amfani da ƙwayar launi na LCCC a lokacin amfani da cutar da za a iya danganta da ciwon sukari, high cholesterol, ko cutar hawan jini.
- Lissafin Cizon Labaran Casa ne ba za ta bi da wani yanayin lafiya ba (kamar cututtukan zuciya, ciwon sukari, hawan jini).
Shawarar ƙwayar ƙwayar ƙwayar ƙwayar ƙwayar ƙwayar ƙwayar ƙwayar cuta (1431697-94-7) Dosage
Lorcaserin HCL foda ya zo a cikin nau'i na kwamfutar hannu kuma ana ɗauka sau 1-2 sau ɗaya a rana, tare da ko ba tare da abinci ba. Dole ne a yi amfani da Lorcaserin tare da rage rage cin abincin kalori da shirin motsa jiki.
The recommended dose of lorcaserin hcl powder is 10 mg administered by mouth twice a day. Lorcaserin may be taken without regard to meals. Lorcaserin hcl should be discontinued in patients who fail to achieve at least a 5% nauyi asara by week 12 since these patients are not likely to experience meaningful weight loss with continued treatment.
Side effects na ƙwayar Lorcaserin Hcl (1431697-94-7)
Lorcaserin Hcl powder is used for the treatment of chronic weight management in adults with a body mass index (BMI) of 30 or greater (obese) as an addition to a reduced-calorie diet and exercise. It is also approved for use by adults with a BMI of 27 or greater (overweight) and who have at least one weight-related condition such as high blood pressure (hypertension), or high cholesterol (dyslipidemia). However, it also may have some illa. As below:
▲ Tshi ne sakamako mafi rinjaye:
- -Bajada,
- -Dizziness,
- -Fatigue,
- -Nausea,
- -Da baki,
- -Constipation, da kuma
- -Hypoglycemia (ƙananan jini sugar).
▲ Other less common but serious illa associated with lorcaserin include:
- -Waɗanda ba a iya amfani da shi ba,
- -Ya canzawa a hankali ko ƙwaƙwalwa,
- -Munanan matsalolin,
- -Depression ko tunani na kashe kansa,
- -Faɗannan abubuwa,
- -Ka sa zuciya,
- -Dajin cikin ƙwayar jini, kuma
- -An karuwa a cikin hormone, prolactin.